Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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106
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106
Tocris Bioscience™ A 410099.1 amide-alkylC4-amine
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IAP ligand with alkyl linker and terminal amine for onward chemistry
107
Tocris Bioscience™ BL660-NO
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Nitric oxide activity-based sensing NIR bioluminescent probe
108
Tocris Bioscience™ AKOS 022
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Voltage-dependent anion channel (VDAC) inhibitor
| Target | Ion Channel Modulators |
|---|---|
| CAS | 878983-38-1 |
| Purity | 0.98 |
| Chemical Name or Material | 1-(4-Chlorophenyl)-3-[4-[[4-(trifluoromethoxy)phenyl]amino]-1-piperidinyl]-2,5-pyrrolidinedione |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H21ClF3N3O3 |
109
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Tocris Bioscience™ AZ 14145845
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Tocris Bioscience™ AZ 14145845
Small and Specialty Supplier Partner
Small and/or specialty supplier based on Federal laws and SBA requirements.
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Small and Specialty Supplier Partner
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Mer/Axl Dual inhibitor
| Target | Additional RTK Inhibitors |
|---|---|
| CAS | 2830555-70-7 |
| Purity | 0.97 |
| Chemical Name or Material | 3-[4-[(Dimethylamino)methyl]phenyl]-N-methyl-N-[5-[3-methyl-5-(1,3,5-trimethyl-1H-pyrazol-4-yl)-2-pyridinyl]-1,3,4-oxadiazol-2-yl]imidazo[1,2-a]pyridine-6-methanamine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C32H35N9O |
110
Tocris Bioscience™ CST 530, Phenol
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Functionalized IAP ligand for PROTACs™
111
Tocris Bioscience™ PRX 07034
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective 5-HT6 receptor antagonist (IC50 = 19 nM, Ki = 4 to 8 nM)
| CAS | 903580-39-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-(1-(5-Chloro-2,3-dimethoxyphenyl)ethyl)-2-(methylsulfonyl)-5-(piperazin-1-yl)aniline hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H28ClN3O4S.HCl |
| Formula Weight | 490.44 |
113
| Shipping Condition | No special requirements |
|---|---|
| CAS | 1441674-54-9 |
| Color | White to Yellow |
| Purity | ≥97.5% |
| Physical Form | Powder |
| Health Hazard 1 | Exclamation mark |
| Chemical Name or Material | Ledipasvir acetone |
| Recommended Storage | Normal conditions |
| Molecular Formula | C49 H54 F2 N8 O6 . C3 H6 O |
| Product Line | Life science |
114
Tocris Bioscience™ AZ1 USP25/28 inhibitor
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective USP25 and USP28 inhibitor
| Target | USP28 |
|---|---|
| CAS | 2165322-94-9 |
| Purity | 0.98 |
| Chemical Name or Material | 2-[[[5-Bromo-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methoxy]phenyl]methyl]amino]ethanol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H16BrF4NO2 |
115
Tocris Bioscience™ AZD 8055
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Highly potent and selective mTOR inhibitor
| Target | mTOR Inhibitors |
|---|---|
| CAS | 1009298-09-2 |
| Purity | 0.98 |
| Chemical Name or Material | 5-[2,4-Bis[(3S)-3-methyl-4-morpholinyl]pyrido[2,3-d]pyrimidin-7-yl]-2-methoxybenzenemethanol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H31N5O4 |
116
Nutlin-3, Thermo Scientific™
CAS: 548472-68-0 Molecular Formula: C30 H30 Cl2 N4 O4 Molecular Weight (g/mol): 581.49 InChI Key: BDUHCSBCVGXTJM-UHFFFAOYNA-N IUPAC Name: 4-[4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazole-1-carbonyl]piperazin-2-one SMILES: COC1=CC=C(C2=NC(C(N2C(=O)N2CCNC(=O)C2)C2=CC=C(Cl)C=C2)C2=CC=C(Cl)C=C2)C(OC(C)C)=C1
| CAS | 548472-68-0 |
|---|---|
| Molecular Weight (g/mol) | 581.49 |
| SMILES | COC1=CC=C(C2=NC(C(N2C(=O)N2CCNC(=O)C2)C2=CC=C(Cl)C=C2)C2=CC=C(Cl)C=C2)C(OC(C)C)=C1 |
| IUPAC Name | 4-[4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazole-1-carbonyl]piperazin-2-one |
| InChI Key | BDUHCSBCVGXTJM-UHFFFAOYNA-N |
| Molecular Formula | C30 H30 Cl2 N4 O4 |
117
Tocris Bioscience™ SLM 6031434 hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective sphingosine kinase 2 (Sphk2) inhibitor
| CAS | 1897379-34-8 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (2S)-2-[3-[4-(Octyloxy)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]-1-pyrrolidinecarboximidamide hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H30F3N5O2.HCl |
118
Tocris Bioscience™ Autophinib
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent VPS34 inhibitor
119
| CAS | 78-44-4 |
|---|---|
| Molecular Formula | C12H24N2O4 |
120
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Thermo Scientific Chemicals Tazarotene
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Thermo Scientific Chemicals Tazarotene
CAS: 118292-40-3 Molecular Formula: C21H21NO2S
| CAS | 118292-40-3 |
|---|---|
| Molecular Formula | C21H21NO2S |